Haridas B Rode
Haridas B Rode
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Chemogenomic profiling provides insights into the limited activity of irreversible EGFR Inhibitors in tumor cells expressing the T790M EGFR resistance mutation
ML Sos, HB Rode, S Heynck, M Peifer, F Fischer, S Klüter, VG Pawar, ...
Cancer research 70 (3), 868-874, 2010
Structure-guided development of affinity probes for tyrosine kinases using chemical genetics
JA Blair, D Rauh, C Kung, CH Yun, QW Fan, H Rode, C Zhang, MJ Eck, ...
Nature Chemical Biology 3 (4), 229-238, 2007
Hybrid compound design to overcome the gatekeeper T338M mutation in cSrc
M Getlik, C Grütter, JR Simard, S Klüter, M Rabiller, HB Rode, ...
Journal of medicinal chemistry 52 (13), 3915-3926, 2009
A new screening assay for allosteric inhibitors of cSrc
JR Simard, S Klüter, C Grütter, M Getlik, M Rabiller, HB Rode, D Rauh
Nature Chemical Biology 5 (6), 394-396, 2009
Structural insights into how irreversible inhibitors can overcome drug resistance in EGFR
A Michalczyk, S Klueter, HB Rode, JR Simard, C Gruetter, M Rabiller, ...
Bioorganic & medicinal chemistry 16 (7), 3482-3488, 2008
Synthesis and biological evaluation of 4-anilinoquinolines as potent inhibitors of epidermal growth factor receptor
VG Pawar, ML Sos, HB Rode, M Rabiller, S Heynck, WAL Van Otterlo, ...
Journal of medicinal chemistry 53 (7), 2892-2901, 2010
Characterization of irreversible kinase inhibitors by directly detecting covalent bond formation: a tool for dissecting kinase drug resistance
S Klüter, JR Simard, HB Rode, C Grütter, V Pawar, HCA Raaijmakers, ...
ChemBioChem 11 (18), 2557-2566, 2010
A chemical genetic approach for covalent inhibition of analogue-sensitive aurora kinase
A Koch, HB Rode, A Richters, D Rauh, S Hauf
ACS chemical biology 7 (4), 723-731, 2012
Analysis of compound synergy in high-throughput cellular screens by population-based lifetime modeling
M Peifer, J Weiss, ML Sos, M Koker, S Heynck, C Netzer, S Fischer, ...
PloS one 5 (1), e8919, 2010
On water direct arylation of imidazo [1, 2-a] pyridines with aryl halides
S Kalari, DA Babar, UB Karale, VB Makane, HB Rode
Tetrahedron Letters 58 (29), 2818-2821, 2017
Synthesis and biological evaluation of 2, 4, 5-trisubstituted thiazoles as antituberculosis agents effective against drug-resistant tuberculosis
UB Karale, VS Krishna, EV Krishna, AS Choudhari, M Shukla, ...
European Journal of Medicinal Chemistry 178, 315-328, 2019
Novel 1, 3, 4-oxadiazoles as antitubercular agents with limited activity against drug-resistant tuberculosis
VB Makane, VS Krishna, EV Krishna, M Shukla, B Mahizhaveni, S Misra, ...
Future Medicinal Chemistry 11 (6), 499-510, 2019
Strategies towards the synthesis of anti-tuberculosis drugs
HB Rode, DM Lade, R Grée, PS Mainkar, S Chandrasekhar
Organic & Biomolecular Chemistry 17 (22), 5428-5459, 2019
Crosslinked enzyme aggregates (CLEA) of phytase with soymilk proteins
H Tirunagari, S Basetty, HB Rode, NW Fadnavis
Journal of biotechnology 282, 67-69, 2018
Identification of new molecular entities (NMEs) as potential leads against tuberculosis from open source compound repository
SS Kotapalli, SSA Nallam, L Nadella, T Banerjee, HB Rode, PS Mainkar, ...
PLoS One 10 (12), e0144018, 2015
Synthesis and evaluation of α-aminoacyl amides as antitubercular agents effective on drug resistant tuberculosis
VB Makane, VS Krishna, EV Krishna, M Shukla, B Mahizhaveni, S Misra, ...
European Journal of Medicinal Chemistry 164, 665-677, 2019
Ligand-free Pd-catalysed decarboxylative arylation of imidazo [1, 2-a] pyridine-3-carboxylic acids with aryl bromides
UB Karale, S Kalari, J Shivakumar, VB Makane, DA Babar, RP Thakare, ...
RSC advances 6 (69), 65095-65104, 2016
Pseudosaccharin amine derivatives: synthesis and elastase inhibitory activity
HB Rode, T Sprang, A Besch, J Loose, HH Otto
Die Pharmazie-An International Journal of Pharmaceutical Sciences 60 (10 …, 2005
A Facile synthesis and antituberculosis properties of almazole D and its enantiomer
DM Lade, VS Krishna, D Sriram, HB Rode
ChemistrySelect 2 (3), 1250-1252, 2017
Synthesis and biological evaluation of 7-substituted-1-(3-bromophenylamino) isoquinoline-4-carbonitriles as inhibitors of myosin light chain kinase and epidermal growth factor …
HB Rode, ML Sos, C Grütter, S Heynck, JR Simard, D Rauh
Bioorganic & medicinal chemistry 19 (1), 429-439, 2011
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