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Sandro Cosconati
Sandro Cosconati
Associate Professor of Medicinal Chemistry, University of Campania "Luigi Vanvitelli"
Verified email at unicampania.it - Homepage
Title
Cited by
Cited by
Year
Virtual screening with AutoDock: theory and practice
S Cosconati, S Forli, AL Perryman, R Harris, DS Goodsell, AJ Olson
Expert opinion on drug discovery 5 (6), 597-607, 2010
5192010
The G‐Triplex DNA
V Limongelli, S De Tito, L Cerofolini, M Fragai, B Pagano, R Trotta, ...
Angewandte Chemie International Edition 52 (8), 2269-2273, 2013
1382013
Identification of 5-arylidene-4-thiazolidinone derivatives endowed with dual activity as aldose reductase inhibitors and antioxidant agents for the treatment of diabetic …
R Ottaną, R Maccari, M Giglio, A Del Corso, M Cappiello, U Mura, ...
European journal of medicinal chemistry 46 (7), 2797-2806, 2011
1152011
Characterizing the 1,4-Dihydropyridines Binding Interactions in the L-Type Ca2+ Channel:  Model Construction and Docking Calculations
S Cosconati, L Marinelli, A Lavecchia, E Novellino
Journal of medicinal chemistry 50 (7), 1504-1513, 2007
1142007
Structural and conformational requisites in DNA quadruplex groove binding: another piece to the puzzle
S Cosconati, L Marinelli, R Trotta, A Virno, S De Tito, R Romagnoli, ...
Journal of the American Chemical Society 132 (18), 6425-6433, 2010
1062010
Sampling protein motion and solvent effect during ligand binding
V Limongelli, L Marinelli, S Cosconati, C La Motta, S Sartini, L Mugnaini, ...
Proceedings of the National Academy of Sciences 109 (5), 1467-1472, 2012
1042012
Tandem application of virtual screening and NMR experiments in the discovery of brand new DNA quadruplex groove binders
S Cosconati, L Marinelli, R Trotta, A Virno, L Mayol, E Novellino, AJ Olson, ...
Journal of the American Chemical Society 131 (45), 16336-16337, 2009
962009
Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells
S Valente, Y Liu, M Schnekenburger, C Zwergel, S Cosconati, C Gros, ...
Journal of medicinal chemistry 57 (3), 701-713, 2014
942014
Design, synthesis, and functionalization of dimeric peptides targeting chemokine receptor CXCR4
O Demmer, I Dijkgraaf, U Schumacher, L Marinelli, S Cosconati, E Gourni, ...
Journal of medicinal chemistry 54 (21), 7648-7662, 2011
922011
Imidazo[2,1-b]thiazole System: A Scaffold Endowing Dihydropyridines with Selective Cardiodepressant Activity
R Budriesi, P Ioan, A Locatelli, S Cosconati, A Leoni, MP Ugenti, ...
Journal of medicinal chemistry 51 (6), 1592-1600, 2008
902008
A balance between elongation and trimming regulates telomere stability in stem cells
T Rivera, C Haggblom, S Cosconati, J Karlseder
Nature structural & molecular biology 24 (1), 30-39, 2017
872017
Conformational Control of Integrin‐Subtype Selectivity in isoDGR Peptide Motifs: A Biological Switch
AO Frank, E Otto, C Mas‐Moruno, HB Schiller, L Marinelli, S Cosconati, ...
Angewandte Chemie International Edition 49 (48), 9278-9281, 2010
872010
Modeling of Cdc25B dual specifity protein phosphatase inhibitors: docking of ligands and enzymatic inhibition mechanism
A Lavecchia, S Cosconati, V Limongelli, E Novellino
ChemMedChem: Chemistry Enabling Drug Discovery 1 (5), 540-550, 2006
752006
Identification of highly conserved residues involved in inhibition of HIV-1 RNase H function by diketo acid derivatives
A Corona, FS Di Leva, S Thierry, L Pescatori, G Cuzzucoli Crucitti, ...
Antimicrobial agents and chemotherapy 58 (10), 6101-6110, 2014
702014
Synthesis, in vitro, and in cell studies of a new series of [indoline-3, 2′-thiazolidine]-based p53 modulators
A Bertamino, M Soprano, S Musella, MR Rusciano, M Sala, E Vernieri, ...
Journal of medicinal chemistry 56 (13), 5407-5421, 2013
692013
Structure-activity relationship of the exopolysaccharide from a psychrophilic bacterium: a strategy for cryoprotection
A Casillo, E Parrilli, F Sannino, DE Mitchell, MI Gibson, G Marino, ...
Carbohydrate polymers 156, 364-371, 2017
622017
A Unique Capsular Polysaccharide Structure from the Psychrophilic Marine Bacterium Colwellia psychrerythraea 34H That Mimics Antifreeze (Glyco)proteins
S Carillo, A Casillo, G Pieretti, E Parrilli, F Sannino, M Bayer-Giraldi, ...
Journal of the American Chemical Society 137 (1), 179-189, 2015
612015
Increasing αvβ3 selectivity of the anti‐angiogenic drug cilengitide by N‐methylation
C Mas‐Moruno, JG Beck, L Doedens, AO Frank, L Marinelli, S Cosconati, ...
Angewandte Chemie International Edition 50 (40), 9496-9500, 2011
612011
Basic quinolinonyl diketo acid derivatives as inhibitors of HIV integrase and their activity against RNase H function of reverse transcriptase
R Costi, M Métifiot, S Chung, G Cuzzucoli Crucitti, K Maddali, L Pescatori, ...
Journal of medicinal chemistry 57 (8), 3223-3234, 2014
582014
Shooting for selective druglike G-quadruplex binders: evidence for telomeric DNA damage and tumor cell death
S Cosconati, A Rizzo, R Trotta, B Pagano, S Iachettini, S De Tito, I Lauri, ...
Journal of medicinal chemistry 55 (22), 9785-9792, 2012
572012
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