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Michael Kassiou
Michael Kassiou
Professor of Medicinal Chemistry, The University of Sydney
Verified email at sydney.edu.au
Title
Cited by
Cited by
Year
Boron in drug discovery: carboranes as unique pharmacophores in biologically active compounds
F Issa, M Kassiou, LM Rendina
Chemical reviews 111 (9), 5701-5722, 2011
6542011
Small animal SPECT and its place in the matrix of molecular imaging technologies
SR Meikle, P Kench, M Kassiou, RB Banati
Physics in Medicine & Biology 50 (22), R45, 2005
4112005
DPA-714, a new translocator protein–specific ligand: Synthesis, radiofluorination, and pharmacologic characterization
ML James, RR Fulton, J Vercoullie, DJ Henderson, L Garreau, S Chalon, ...
Journal of Nuclear Medicine 49 (5), 814-822, 2008
2862008
Molecular imaging of microglial activation in amyotrophic lateral sclerosis
P Corcia, C Tauber, J Vercoullie, N Arlicot, C Prunier, J Praline, G Nicolas, ...
PloS one 7 (12), e52941, 2012
2732012
Comparative evaluation of the translocator protein radioligands 11C-DPA-713, 18F-DPA-714, and 11C-PK11195 in a rat model of acute neuroinflammation
F Chauveau, N Van Camp, F Dollé, B Kuhnast, F Hinnen, A Damont, ...
Journal of Nuclear Medicine 50 (3), 468-476, 2009
2632009
Neuroinflammation and brain atrophy in former NFL players: an in vivo multimodal imaging pilot study
JM Coughlin, Y Wang, CA Munro, S Ma, C Yue, S Chen, R Airan, PK Kim, ...
Neurobiology of disease 74, 58-65, 2015
2512015
Pharmacology of Valinate and tert-Leucinate Synthetic Cannabinoids 5F-AMBICA, 5F-AMB, 5F-ADB, AMB-FUBINACA, MDMB-FUBINACA, MDMB-CHMICA, and …
SD Banister, M Longworth, R Kevin, S Sachdev, M Santiago, J Stuart, ...
ACS Chemical Neuroscience 7 (9), 1241-1254, 2016
2472016
Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists
A Gillis, AB Gondin, A Kliewer, J Sanchez, HD Lim, C Alamein, ...
Science signaling 13 (625), eaaz3140, 2020
2422020
Brain inflammation is induced by co-morbidities and risk factors for stroke
C Drake, H Boutin, MS Jones, A Denes, BW McColl, JR Selvarajah, ...
Brain, behavior, and immunity 25 (6), 1113-1122, 2011
2342011
Pharmacology of indole and indazole synthetic cannabinoid designer drugs ab-fubinaca, adb-fubinaca, ab-pinaca, adb-pinaca, 5f-ab-pinaca, 5f-adb-pinaca, adbica, and 5f-adbica
SD Banister, M Moir, J Stuart, RC Kevin, KE Wood, M Longworth, ...
ACS chemical neuroscience 6 (9), 1546-1559, 2015
2282015
Effects of bioisosteric fluorine in synthetic cannabinoid designer drugs JWH-018, AM-2201, UR-144, XLR-11, PB-22, 5F-PB-22, APICA, and STS-135
SD Banister, J Stuart, RC Kevin, A Edington, M Longworth, SM Wilkinson, ...
ACS Chemical Neuroscience 6 (8), 1445-1458, 2015
2072015
Evaluation of the PBR/TSPO Radioligand [18F]DPA-714 in a Rat Model of Focal Cerebral Ischemia
A Martín, R Boisgard, B Thézé, N Van Camp, B Kuhnast, A Damont, ...
Journal of Cerebral Blood Flow & Metabolism 30 (1), 230-241, 2010
2002010
Translational evaluation of translocator protein as a marker of neuroinflammation in schizophrenia
T Notter, JM Coughlin, T Gschwind, U Weber-Stadlbauer, Y Wang, ...
Molecular psychiatry 23 (2), 323-334, 2018
1982018
The translocator protein
AM Scarf, M Kassiou
Journal of Nuclear Medicine 52 (5), 677-680, 2011
1942011
Recent developments in TSPO PET imaging as a biomarker of neuroinflammation in neurodegenerative disorders
EL Werry, FM Bright, O Piguet, LM Ittner, GM Halliday, JR Hodges, ...
International journal of molecular sciences 20 (13), 3161, 2019
1932019
Neuroinflammation in frontotemporal dementia
F Bright, EL Werry, C Dobson-Stone, O Piguet, LM Ittner, GM Halliday, ...
Nature Reviews Neurology 15 (9), 540-555, 2019
1922019
11C-DPA-713: a novel peripheral benzodiazepine receptor PET ligand for in vivo imaging of neuroinflammation
H Boutin, F Chauveau, C Thominiaux, MC Grégoire, ML James, ...
Journal of Nuclear Medicine 48 (4), 573-581, 2007
1772007
Developing a preclinical model of Parkinson's disease: a study of behaviour in rats with graded 6-OHDA lesions
L Truong, H Allbutt, M Kassiou, JM Henderson
Behavioural brain research 169 (1), 1-9, 2006
1732006
An overview of late-stage functionalization in today’s drug discovery
M Moir, JJ Danon, TA Reekie, M Kassiou
Expert opinion on drug discovery 14 (11), 1137-1149, 2019
1662019
Positron emission tomography imaging of neuroinflammation
A Cagnin, M Kassiou, SR Meikle, RB Banati
Neurotherapeutics 4, 443-452, 2007
1642007
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