| Quantitative live-cell kinetic degradation and mechanistic profiling of PROTAC mode of action KM Riching, S Mahan, CR Corona, M McDougall, JD Vasta, MB Robers, ... ACS chemical biology 13 (9), 2758-2770, 2018 | 224 | 2018 |
| Quantitative, wide-spectrum kinase profiling in live cells for assessing the effect of cellular ATP on target engagement JD Vasta, CR Corona, J Wilkinson, CA Zimprich, JR Hartnett, MR Ingold, ... Cell chemical biology 25 (2), 206-214. e11, 2018 | 213 | 2018 |
| Synthetic estrogen derivatives demonstrate the functionality of intracellular GPR30 CM Revankar, HD Mitchell, AS Field, R Burai, C Corona, C Ramesh, ... ACS Chemical Biology 2 (8), 536-544, 2007 | 207 | 2007 |
| Selective JAK3 inhibitors with a covalent reversible binding mode targeting a new induced fit binding pocket M Forster, A Chaikuad, SM Bauer, J Holstein, MB Robers, CR Corona, ... Cell chemical biology 23 (11), 1335-1340, 2016 | 108 | 2016 |
| Discovery of a selective inhibitor of doublecortin like kinase 1 FM Ferguson, B Nabet, S Raghavan, Y Liu, AL Leggett, M Kuljanin, ... Nature chemical biology 16 (6), 635-643, 2020 | 92 | 2020 |
| Bisphenol A directly targets tubulin to disrupt spindle organization in embryonic and somatic cells O George, BK Bryant, R Chinnasamy, C Corona, JB Arterburn, ... ACS chemical biology 3 (3), 167-179, 2008 | 86 | 2008 |
| Quantifying CDK inhibitor selectivity in live cells CI Wells, JD Vasta, CR Corona, J Wilkinson, CA Zimprich, MR Ingold, ... Nature communications 11 (1), 2743, 2020 | 78 | 2020 |
| Synthesis of 17-α-Substituted Estradiol-Pyridin-2-yl Hydrazine Conjugates as Effective Ligands for Labeling with Alberto's Complex fac-[Re(OH2)3(CO)3]+ in … JB Arterburn, C Corona, KV Rao, KE Carlson, JA Katzenellenbogen The Journal of Organic Chemistry 68 (18), 7063-7070, 2003 | 69 | 2003 |
| In Vivo Stable Tumor-Specific Painting in Various Colors Using Dehalogenase-Based Protein-Tag Fluorescent Ligands N Kosaka, M Ogawa, PL Choyke, N Karassina, C Corona, M McDougall, ... Bioconjugate chemistry 20 (7), 1367-1374, 2009 | 63 | 2009 |
| Synthesis of a biotin-derived alkyne for Pd-catalyzed coupling reactions C Corona, BK Bryant, JB Arterburn Organic letters 8 (9), 1883-1886, 2006 | 63 | 2006 |
| KRAS is vulnerable to reversible switch-II pocket engagement in cells JD Vasta, DM Peacock, Q Zheng, JA Walker, Z Zhang, CA Zimprich, ... Nature chemical biology 18 (6), 596-604, 2022 | 57 | 2022 |
| Homogeneous plate based antibody internalization assay using pH sensor fluorescent dye N Nath, B Godat, C Zimprich, SJ Dwight, C Corona, M McDougall, M Urh Journal of immunological methods 431, 11-21, 2016 | 55 | 2016 |
| Quantitative, real-time measurements of intracellular target engagement using energy transfer MB Robers, JD Vasta, CR Corona, RF Ohana, R Hurst, MA Jhala, ... Systems Chemical Biology: Methods and Protocols, 45-71, 2019 | 46 | 2019 |
| Proluciferin acetals as bioluminogenic substrates for cytochrome P450 activity and probes for CYP3A inhibition PL Meisenheimer, HT Uyeda, D Ma, M Sobol, MG McDougall, C Corona, ... Drug metabolism and disposition 39 (12), 2403-2410, 2011 | 38 | 2011 |
| NanoClick: a high throughput, target-agnostic peptide cell permeability assay A Peier, L Ge, N Boyer, J Frost, R Duggal, K Biswas, S Edmondson, ... ACS Chemical Biology 16 (2), 293-309, 2021 | 36 | 2021 |
| A luminescent assay for real-time measurements of receptor endocytosis in living cells MB Robers, BF Binkowski, M Cong, C Zimprich, C Corona, M McDougall, ... Analytical biochemistry 489, 1-8, 2015 | 24 | 2015 |
| Design of a “two-in-one” mutant-selective epidermal growth factor receptor inhibitor that spans the orthosteric and allosteric sites F Wittlinger, DE Heppner, C To, M Günther, BH Shin, JK Rana, ... Journal of Medicinal Chemistry 65 (2), 1370-1383, 2021 | 18 | 2021 |
| A Toolbox for the Generation of Chemical Probes for Baculovirus IAP Repeat Containing Proteins MP Schwalm, LM Berger, MN Meuter, JD Vasta, CR Corona, S Röhm, ... Frontiers in Cell and Developmental Biology 10, 2022 | 12 | 2022 |
| A high-throughput method to prioritize PROTAC intracellular target engagement and cell permeability using NanoBRET JD Vasta, CR Corona, MB Robers Targeted Protein Degradation: Methods and Protocols, 265-282, 2021 | 12 | 2021 |
| Luminogenic compounds and methods to detect cytochrome P450 3A enzymes C Corona, P Meisenheimer, HT Uyeda US Patent 8,288,559, 2012 | 11 | 2012 |
